- Drug Class: Aromatase Inhibitor
- Active substance: Exemestane 25 mg
- Active half-life: 9 Hours
- Dosage: 12.5-25 mg/day
- Acne: No
- Hepatotoxicity: No
- Aromatization: No
- Manufacturer: Dragon Pharma
- Listed: May 5, 2017 11:13 am
- Expires: 8557 days, 21 hours
In medicine, such a hormonal agent can be effectively used as an antiestrogenic antitumor drug. In sports practice, it is usually used as an aid in courses of aromatized AAS (for the prevention or elimination of estrogenic side effects, in particular gynecomastia).
The active substance of this drug, Exemestane, is a strong steroidal antiestrogen with the ability to block the enzyme aromatase (belongs to the third generation of aromatase inhibitors). Exemestane was created exclusively for medical use, in particular for the treatment of neoplastic diseases.
If you give a description specifically to Aromasin by Dragon Pharma, then to begin with it is worth noting that the drug, when properly applied, is able to exert a pronounced antitumoral, anti-estrogenic effect. It inhibits aromatase by irreversible binding to the active center of the enzyme, which causes its inactivation, and blocks the formation of estrogens. That is important, thus it does not show estrogenic or progestogenic activity and does not influence synthesis of a cortisol and aldosterone in adrenals.
The action of Aromasin also increases the levels of LH (luteinizing hormone) and FSH (follicle-stimulating hormone) due to feedback, when a decrease in the concentration of estrogens leads to an increase in the level of gonadotropins. LH and FSH, among other things, are necessary for the correct operation of the reproductive system and the synthesis of Testosterone (LH is able to stimulate Leydig interstitial cells producing testosterone).
It is important to clarify that Aromasin tablets manufactured by Dragon Pharmaceuticals cause a direct dose-dependent reduction in the content of estradiol, estrone and estrone sulfate. It should also be mentioned that they may have a slight androgenic activity.
Aromasin Dosage / Cycle / Stack
In sports practice, in particular in bodybuilding, this anti-estrogenic drug is taken predominantly by men. It is usually used during heavy steroid courses of flavoring steroids to block the process of aromatization and certainly to protect against the occurrence of associated side effects (gynecomastia in men, excessive water retention, increase in fat layer).
How to use Aromasin from Dragon Pharma? If the drug is used to prevent estrogenic side effects during the course, then dosage should be used around 12.5 mg per day or 25 mg in 1-2 days (respectively, half a tablet a day or a whole tablet every 2-3 days). If the reception begins already with the appearance of side effects, then the dosage should be higher – around 25 mg per day (ie 1 tablet a day).
After the use of Aromasin, the active ingredient quickly takes over the case. At reception after meal Cmax in a blood is reached within only two hours. By the way, food intake is able to improve better absorption (the reached level of absorption after eating is 40% higher than when applied on an empty stomach). And this means that you should drink tablets after eating, and not on an empty stomach.
Instructions for Aromasin use: You are unlikely to say this, but the drug is output, as it does, usually quite quickly. More specifically, after a single dose, excretion takes place on an average of 1 week (with urine and feces in equal parts).
What are the contraindications for the use of this antiestrogenic agent? First of all it is hypersensitivity to the active substance or components in the composition. In addition, the drug is contraindicated in childhood and women during pregnancy and lactation.
Aromasin Side Effects
Can an athlete who uses Aromasin (Exemestane) in tablets worry about side effects and if so, which ones? When taking moderate doses, the risk of side effects is low, but in some cases, certain abnormalities can still occur. For example, you can be told about yourself such sides as headaches, dizziness, nausea, constipation, increased sweating and even sleep disorders.
What are the storage conditions? Here everything is simple: first, do not subject the drug to sudden temperature changes and keep it in a dark and dry place; Secondly, the storage temperature is usually recommended room temperature, do not forget about it.
In general, Aromasin 25mg is a strong enough and effective antiestrogenic agent (aromatase inhibitor), the reviews of which serve as confirmation of this fact. It is an excellent aromatase inhibitor and an analogue of Anastrozole.
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