Tamoxifen is a competitive inhibitor of peripheral estrogen receptor. And if earlier it was believed that the drug does not have the influence of estrogen, but today this view is completely rejected. In fact, the ratio of agonist and antagonist activity equal to 45/55. Chemically Tamoxifen is a derivative form of triphenylethylene. The drug belongs to the group of sex hormones. Initially it was used for the treatment of cancers in women (breast cancer). But, undoubtedly, today Tamoxifen is much more common in the field of sports and bodybuilding in particular.
Tamoxifen Citrate for Bodybuilding
It is no secret that the majority of aromatazing steroids are exposed, that is to be converted in the female sex hormones - estrogens. This can lead to a variety of side effects which can be combated using Tamoxifen. Unlike other means of such effects, the substance is neither androgen or anabiotic.
- Increase in power rates.
- Increased hardness and muscle relief.
- The growth of muscle mass. Bodybuilders buy Tamoxifen, which is very popular in bodybuilding, argued that without it can not do any one victory in major competitions.
- Marked anti-estrogen effects. The effect that has made so popular Tamoxifen for sale. The higher dosage of AAS, the need for large compensation estrogenic activity. The use of Tamoxifen or analogues thereof at PCT after heavy cycles is virtually mandatory.
- Fighting fat deposits.
- Prevention of feminization.
- Reducing the risk of atherosclerosis, the prevention of cardiovascular disease.
- Improving liver.
Tamoxifen's antiestrogen effects are caused by blocking the estrogen receptors (but not the termination of the conversion of testosterone to estrogen, as many think). The drug only freezes estrogenic activity but does not prevent it entirely.
Tamoxifen Dosage / Tamoxifen Post Cycle Therapy
Tamoxifen after a cycle of steroids should be combined with aromatase inhibitors, the most popular of which is Proviron (it is often used for the reason that it does not inhibit the production of growth hormone and inhibits aromatase, thereby increasing the concentration of anabolic hormones in the blood). Tamoxifen as a primary means for Post Cycle Therapy is used in dosages of 10 to 20 milligrams daily, starting from the last week of the cycle and ending with the second week after its completion. If Proviron is not accepted, Tamoxifen is included later - at 2 weeks and ends 2-3 weeks after its cancellation.
Tamoxifen Side Effects
The most common side effects of Tamoxifen are associated with its pronounced antiestrogenic properties. Exceeding the recommended dose and/or duration of the cycle can cause in female: hair loss or even complete hair loss, flushing intense heat, itching in the crotch area, pain in the bones; male - fever, dizziness, nausea. Due to the water retention disrupt the normal functioning of the kidneys. Also, sometimes there are bouts of depression, depression and drowsiness. Excessive intake is fraught with fatigue, constipation and anorexia. You may experience inflammation of the retina, cataract, partial or complete loss of vision. Tamoxifen is sometimes accompanied by a rash on the skin. Cases of occurrence of headaches, changes in the cornea, confusion of consciousness. Liver disorders occur only in case of serious diseases of the body (such as hepatitis).
Note that the highest levels of estrogen in the body is observed at the end of the first week of the AAS cycle. As for how to take Tamoxifen in bodybuilding on a cycle of steroids, which has no flavoring effect, it is recommended to add it only at the end of the cycle.
It is often expressed about the preparation not by athletes, as Tamoxifen for many years have been used in post-menopausal women with estrogen-receptor-positive patients and breast cancer. As for the athletes, they noted a pronounced anti-estrogen effects. Despite the wide range of possible side effects of Tamoxifen, reviews indicate that adverse reactions are extremely rare.
Women athletes talk about the inability to use the drug during pregnancy. Moreover, it can inhibit ovum implantation in the uterine wall. Reviews of Tamoxifen on the entry-level athletes are rare because amateurs are often bypassed by simple solo AAS cycles that do not require PCT.